SCHEMBL4724929

SCHEMBL4724929

CNC(=O)CCCNc1ccc(C(F)(F)F)c(-n2nc(-c3cc(OC)cc(OC)c3)c3c(c2=O)NCC3)c1

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SCD O00767 3/20 0.32
FPR1 P21462 1/20 0.31
FPR2 P25090 1/20 0.31
NTRK1 P04629 1/20 0.31
BRAF P15056 1/20 0.31
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30
KMT2A Q03164 2/20 0.30
KDM4E B2RXH2 1/20 0.30
HSD17B1 P14061 1/20 0.30
HSD17B2 P37059 1/20 0.30
EPHX2 P34913 1/20 0.30
MEN1 O00255 1/20 0.30
EHMT2 Q96KQ7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4724753 0.90 BRAF (0.33) SCDNTRK1BRAFHTR2CHTR2B
SCHEMBL4723187 0.88 MAPT (0.34) SCDFPR1FPR2KMT2AKDM4E
SCHEMBL4719384 0.86 MAPT (0.34) SCDFPR1FPR2KMT2AKDM4E
SCHEMBL4722630 0.84 F10 (0.31) SCDFPR1FPR2KMT2AKDM4E
SCHEMBL4719755 0.83 MAPT (0.35) SCDFPR1FPR2KMT2AKDM4E
SCHEMBL4719300 0.82 BRD4 (0.35) SCDFPR1FPR2HSD17B1HSD17B2
SCHEMBL4720527 0.82 SCD (0.34) SCDFPR1FPR2KDM4EHSD17B1
SCHEMBL4765721 0.80 PDE4A (0.36) SCDKMT2AKDM4EMEN1
SCHEMBL4719449 0.80 PDE4A (0.36) SCDKMT2AKDM4EMEN1
SCHEMBL4720876 0.80 CYP11B1 (0.33) NTRK1HTR2CHTR2BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed