SCHEMBL4720727

SCHEMBL4720727

NC(=O)[C@H]1CCCCN1C1CCN(C(=O)[CH]Cc2cc(Cl)c(N)c(C(F)(F)F)c2)CC1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.37
TACR2 P21452 1/20 0.35
TACR1 P25103 1/20 0.35
RAMP1 O60894 1/20 0.35
CALCRL Q16602 1/20 0.35
RORC P51449 1/20 0.32
WNT3 P56703 1/20 0.32
SFRP1 Q8N474 1/20 0.32
KRAS P01116 1/20 0.31
EPHX1 P07099 1/20 0.30
NOTUM Q6P988 1/20 0.30
ENPP2 Q13822 1/20 0.30
XIAP P98170 1/20 0.30
LRRK2 Q5S007 1/20 0.30
EPHX2 P34913 1/20 0.30
SLC9A1 P19634 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4718767 1.00 ADRB2 (0.37) ADRB2TACR2TACR1RAMP1CALCRL
SCHEMBL5248989 0.81 RAMP1 (0.42) ADRB2RAMP1CALCRLENPP2LRRK2
SCHEMBL4849662 0.81 RAMP1 (0.41) ADRB2RAMP1CALCRLNOTUMLRRK2
SCHEMBL4720816 0.79 RAMP1 (0.35) ADRB2TACR1RAMP1CALCRLRORC
SCHEMBL4804839 0.77 TEAD1 (0.39) ADRB2RAMP1CALCRLEPHX2
SCHEMBL5326014 0.74 ACACB (0.35) RAMP1CALCRLSLC9A1
SCHEMBL4798589 0.73 TEAD1 (0.36) ADRB2RAMP1CALCRLEPHX2
SCHEMBL3593151 0.70 CNR2 (0.30)
SCHEMBL4763044 0.70 NOTUM (0.34) KRASNOTUM
SCHEMBL8190796 0.69 SPHK1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558600-B1 SELECTED CGRP ANTAGONISTS, METHOD FOR PRODUCTION AND USE THEREOF AS MEDICAMENT BOEHRINGER INGELHEIM PHARMA (DE) 2008-05-07 EP claimed