SCHEMBL4720740

SCHEMBL4720740

COc1cc(OC)cc(-c2nn(-c3cc(NC4CC4)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
GRM7 Q14831 1/20 0.34
CNR2 P34972 3/20 0.34
CNR1 P21554 1/20 0.34
AR P10275 4/20 0.33
UGCG Q16739 1/20 0.32
ULK1 O75385 2/20 0.32
ULK2 Q8IYT8 2/20 0.32
HRH3 Q9Y5N1 1/20 0.32
F10 P00742 1/20 0.32
GFER P55789 1/20 0.32
PABPC1 P11940 1/20 0.32
SMURF1 Q9HCE7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4719123 0.97 AR (0.37) PDE4APDE4BPDE4CPDE4DGRM7
SCHEMBL4720922 0.89 F10 (0.39) PDE4APDE4BPDE4CPDE4DGRM7
SCHEMBL4722944 0.88 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DGRM7
SCHEMBL4724950 0.87 UTS2R (0.36) PDE4APDE4BPDE4CPDE4DGRM7
SCHEMBL4724044 0.87 CNR2 (0.39) PDE4APDE4BPDE4CPDE4DGRM7
SCHEMBL4720454 0.87 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DGRM7
SCHEMBL4724087 0.86 UTS2R (0.35) PDE4APDE4BPDE4CPDE4DGRM7
SCHEMBL4723085 0.86 CNR2 (0.37) PDE4APDE4BPDE4CPDE4DGRM7
SCHEMBL4721150 0.86 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DGRM7
SCHEMBL4722165 0.86 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed