SCHEMBL4722165

SCHEMBL4722165

COc1cc(OC)cc(-c2nn(-c3cc(Nc4ccccc4)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.43
PDE4B Q07343 2/20 0.43
PDE4C Q08493 2/20 0.43
PDE4D Q08499 2/20 0.43
CNR2 P34972 5/20 0.40
CNR1 P21554 2/20 0.40
MAPT P10636 4/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
MAPK1 P28482 2/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MAPK14 Q16539 2/20 0.35
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720922 0.89 F10 (0.39) PDE4APDE4BPDE4CPDE4DCNR2
SCHEMBL4721038 0.88 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL4722944 0.88 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DCNR2
SCHEMBL4724135 0.88 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL4722274 0.87 PDE4A (0.48) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL4720454 0.87 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DCNR2
SCHEMBL4720114 0.86 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DCNR2
SCHEMBL4721150 0.86 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL4721102 0.86 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DCNR2
SCHEMBL4724043 0.86 F10 (0.42) PDE4APDE4BPDE4CPDE4DMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed