SCHEMBL4721776

SCHEMBL4721776

CCCCNS(=O)(=O)c1ccc(B2OC(C)(C)C(C)(C)O2)s1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
HTT P42858 2/20 0.50
TSHR P16473 2/20 0.50
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 4/20 0.40
MAPK1 P28482 1/20 0.38
LPL P06858 5/20 0.36
LIPG Q9Y5X9 5/20 0.36
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
LMNA P02545 2/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
ALOX12 P18054 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
RECQL P46063 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1164818 0.84 ALDH1A1 (0.45) KMT2ASMN1; SMN2HTTTSHRMEN1
SCHEMBL1164490 0.84 KMT2A (0.48) KMT2ASMN1; SMN2HTTTSHRMEN1
SCHEMBL12846047 0.81 MAPK1 (0.42) KMT2ASMN1; SMN2HTTTSHRMEN1
SCHEMBL1164297 0.79 CA1 (0.38) SMN1; SMN2LPLLIPGCA12CA9
SCHEMBL16004583 0.79 ALDH1A1 (0.33) KMT2ASMN1; SMN2HTTTSHRMEN1
SCHEMBL1164423 0.79 SMN1; SMN2 (0.34) KMT2ASMN1; SMN2HTTTSHRMEN1
SCHEMBL1163931 0.79 CA1 (0.35) KMT2ASMN1; SMN2HTTMEN1ALDH1A1
SCHEMBL1164320 0.74 LOX (0.39) LPLLIPGCA12CA9
SCHEMBL11051510 0.73 KMT2A (0.61) KMT2ASMN1; SMN2HTTTSHRMEN1
SCHEMBL2288390 0.73 CA12 (0.51) KMT2ASMN1; SMN2HTTTSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001849-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS F. Hoffmann-Roche AG (CH) 2008-12-17 EP disclosed
WO-2007110337-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2007-10-04 WO disclosed