SCHEMBL4721956

SCHEMBL4721956

COc1cc(OC)cc(-c2nn(-c3cc(N4CC[C@H](OC)C4)ccc3C(F)(F)F)c(=O)c3c2CCN3CCO)c1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACACB O00763 3/20 0.34
KDM1A O60341 6/20 0.33
F10 P00742 5/20 0.32
F2 P00734 1/20 0.32
IDH1 O75874 2/20 0.31
S1PR1 P21453 1/20 0.31
FFAR1 O14842 1/20 0.31
CXCR3 P49682 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4721962 1.00 ACACB (0.34) ACACBKDM1AF10F2IDH1
SCHEMBL4721691 0.92 F10 (0.38) F10F2
SCHEMBL4721689 0.92 F10 (0.38) F10F2
SCHEMBL4724293 0.92 F10 (0.38) F10F2
SCHEMBL4721664 0.90 F10 (0.35) F10F2CXCR3
SCHEMBL4723157 0.89 F10 (0.32) F10F2CXCR3
SCHEMBL4724288 0.89 F10 (0.40) F10F2
SCHEMBL4722374 0.88 ITGB2 (0.37) ACACBF10
SCHEMBL4722251 0.88 ITGB2 (0.37) ACACBF10
SCHEMBL4766491 0.88 ITGB2 (0.37) ACACBF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed