SCHEMBL4722089

SCHEMBL4722089

COc1cc(OC)cc(-c2nn(-c3cc(NCCO)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
SCD O00767 3/20 0.35
MAPT P10636 3/20 0.34
SMN1; SMN2 Q16637 4/20 0.33
CNR2 P34972 3/20 0.33
TP53 P04637 1/20 0.33
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
KDM4E B2RXH2 1/20 0.33
TSHR P16473 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
CNR1 P21554 1/20 0.32
F10 P00742 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4719833 0.95 PDE4A (0.35) PDE4APDE4BPDE4CPDE4DSCD
SCHEMBL4722084 0.94 PDE4A (0.35) PDE4APDE4BPDE4CPDE4DSCD
SCHEMBL4721220 0.93 PDE4A (0.35) PDE4APDE4BPDE4CPDE4DSCD
SCHEMBL4721102 0.92 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DSCD
SCHEMBL14101739 0.91 PDE4A (0.36) PDE4APDE4BPDE4CPDE4DSCD
SCHEMBL14101915 0.91 PDE4A (0.36) PDE4APDE4BPDE4CPDE4DSCD
SCHEMBL4720454 0.91 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DSCD
SCHEMBL4722572 0.91 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DSCD
SCHEMBL4723445 0.91 SMN1; SMN2 (0.35) PDE4APDE4BPDE4CPDE4DSCD
Hydrochloric Acid SCHEMBL4720194 0.91 PDE4A (0.36) PDE4APDE4BPDE4CPDE4DSCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed