SCHEMBL4722572

SCHEMBL4722572

COc1cc(OC)cc(-c2nn(-c3cc(NCCC(=O)O)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
S1PR1 P21453 1/20 0.36
MAPT P10636 4/20 0.36
SMN1; SMN2 Q16637 4/20 0.35
TP53 P04637 2/20 0.35
ALDH1A1 P00352 2/20 0.34
SCD O00767 1/20 0.34
GCGR P47871 1/20 0.34
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
GAA P10253 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4719449 0.95 PDE4A (0.36) PDE4APDE4BPDE4CPDE4DS1PR1
SCHEMBL4723364 0.94 PDE4A (0.35) PDE4APDE4BPDE4CPDE4DS1PR1
SCHEMBL4723445 0.93 SMN1; SMN2 (0.35) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL4722266 0.93 PDE4A (0.36) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL4723112 0.93 PDE4A (0.39) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL4721347 0.92 PDE4A (0.34) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL4719755 0.92 MAPT (0.35) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL4722089 0.91 PDE4A (0.36) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL4765721 0.90 PDE4A (0.36) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL4721102 0.90 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed