SCHEMBL4722110

SCHEMBL4722110

N#Cc1cc(N2CCC(O)C2)ccc1C(F)(F)F

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AR P10275 7/20 0.62
NOTUM Q6P988 8/20 0.45
HSD11B1 P28845 3/20 0.40
CDK1 P06493 1/20 0.40
CDK2 P24941 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722109 1.00 AR (0.62) ARNOTUMHSD11B1CDK1CDK2
SCHEMBL15564231 0.81 AR (0.64) AR
SCHEMBL2935853 0.81 NOTUM (0.49) ARNOTUMHSD11B1CDK1CDK2
SCHEMBL15938046 0.80 AR (0.67) ARNOTUMCDK1CDK2
SCHEMBL16071294 0.80 AR (0.67) ARNOTUMCDK1CDK2
SCHEMBL15938045 0.80 AR (0.67) ARNOTUMCDK1CDK2
SCHEMBL4723399 0.80 NOTUM (0.48) ARNOTUMHSD11B1CDK1CDK2
SCHEMBL4723392 0.80 NOTUM (0.48) ARNOTUMHSD11B1CDK1CDK2
SCHEMBL1409422 0.78 NOTUM (0.67) ARNOTUMHSD11B1
SCHEMBL13651213 0.77 AR (1.00) ARNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed