SCHEMBL4723399

SCHEMBL4723399

OC1CCN(c2ccc(C(F)(F)F)c(Br)c2)C1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 10/20 0.48
AR P10275 1/20 0.46
CDK1 P06493 1/20 0.42
CDK2 P24941 1/20 0.42
HSD11B1 P28845 3/20 0.41
SOS1 Q07889 2/20 0.41
P2RX7 Q99572 1/20 0.41
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4723392 1.00 NOTUM (0.48) NOTUMARCDK1CDK2HSD11B1
SCHEMBL2935853 0.84 NOTUM (0.49) NOTUMARCDK1CDK2HSD11B1
SCHEMBL1409422 0.81 NOTUM (0.67) NOTUMARHSD11B1
SCHEMBL4721681 0.80 NOTUM (0.44) NOTUMARCDK1CDK2HSD11B1
SCHEMBL2050734 0.80 NOTUM (0.49) NOTUMARCDK1CDK2HSD11B1
SCHEMBL2050735 0.80 NOTUM (0.49) NOTUMARCDK1CDK2HSD11B1
SCHEMBL1409621 0.80 NOTUM (0.68) NOTUMAR
SCHEMBL2971480 0.80 NOTUM (0.49) NOTUMARCDK1CDK2HSD11B1
SCHEMBL4722110 0.80 AR (0.62) NOTUMARCDK1CDK2HSD11B1
SCHEMBL4722109 0.80 AR (0.62) NOTUMARCDK1CDK2HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed