SCHEMBL4722596

SCHEMBL4722596

CC[C@@H](N)C1(C)N=CC(c2ccc(C[C@@H](CCO)NC(=O)c3ccc(OC(C)C)c(Cl)c3)cc2)=N1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CENPE Q02224 3/20 0.43
KIFC1 Q9BW19 1/20 0.39
TAS1R3 Q7RTX0 4/20 0.37
TAS1R1 Q7RTX1 4/20 0.37
ROCK2 O75116 1/20 0.35
PRKACA P17612 1/20 0.35
RPS6KB1 P23443 1/20 0.35
IRAK1 P51617 1/20 0.35
PRKX P51817 1/20 0.35
LIMK1 P53667 1/20 0.35
PRKG2 Q13237 1/20 0.35
ROCK1 Q13464 1/20 0.35
PRKG1 Q13976 1/20 0.35
PKN2 Q16513 1/20 0.35
HIPK4 Q8NE63 1/20 0.35
AURKB Q96GD4 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
CSNK1G1 Q9HCP0 1/20 0.35
S1PR1 P21453 3/20 0.33
RAB9A P51151 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4774113 0.77 CENPE (0.54) CENPEKIFC1TAS1R3TAS1R1ROCK2
SCHEMBL3229399 0.76 CENPE (0.52) CENPEKIFC1TAS1R3TAS1R1ROCK2
SCHEMBL2106289 0.76 CENPE (0.53) CENPEKIFC1TAS1R3TAS1R1ROCK2
SCHEMBL3233445 0.75 CENPE (0.52) CENPEKIFC1TAS1R3TAS1R1ROCK2
SCHEMBL13711223 0.75 CENPE (0.54) CENPEKIFC1TAS1R3TAS1R1ROCK2
SCHEMBL2617412 0.75 CENPE (0.54) CENPEKIFC1TAS1R3TAS1R1ROCK2
SCHEMBL2104926 0.74 CENPE (0.56) CENPEKIFC1TAS1R3TAS1R1S1PR1
SCHEMBL13626726 0.74 CENPE (0.53) CENPEKIFC1TAS1R3TAS1R1ROCK2
SCHEMBL2101923 0.73 CENPE (0.51) CENPETAS1R3TAS1R1ROCK2PRKACA
SCHEMBL3469159 0.73 CENPE (0.51) CENPETAS1R3TAS1R1ROCK2PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951719-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-08-06 EP disclosed
WO-2007056469-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO disclosed