SCHEMBL4722607

SCHEMBL4722607

CCCCCN(C)c1ccc(N(C(N)=O)c2nc(-c3ccc(C)nc3)cs2)cc1C(F)(F)F.CCCCOc1ccc(N(C(N)=O)c2nc(-c3ccc(F)c(F)c3)cs2)cc1C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34
NR1H2 P55055 3/20 0.33
PPARD Q03181 3/20 0.33
PPARA Q07869 3/20 0.33
NR1H3 Q13133 3/20 0.33
S1PR1 P21453 5/20 0.33
S1PR4 O95977 3/20 0.33
S1PR5 Q9H228 3/20 0.33
MEN1 O00255 2/20 0.33
RAB9A P51151 2/20 0.33
KMT2A Q03164 2/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
NFKB1 P19838 1/20 0.33
MAPK1 P28482 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5423224 0.90 PDE3B (0.36) NPC1MAPK14ATP4AATP4B
SCHEMBL23553880 0.90 NR1H2 (0.35) THRATHRBNR1H2PPARDPPARA
SCHEMBL9101422 0.89 MAPK14 (0.37) PPARAMEN1RAB9AKMT2APPARG
SCHEMBL5430460 0.88 NPC1 (0.39) THRATHRBPPARDS1PR1S1PR4
SCHEMBL5428996 0.88 MEN1 (0.41) THRATHRBS1PR1S1PR4S1PR5
SCHEMBL4656403 0.82 MAPK14 (0.46) MEN1RAB9AKMT2ANPC1ALDH1A1
SCHEMBL4655528 0.81 THRA (0.41) THRATHRBNR1H2PPARDPPARA
SCHEMBL9098567 0.81 S1PR4 (0.40) THRATHRBS1PR1S1PR4S1PR5
SCHEMBL4656609 0.81 MAPK14 (0.47) THRATHRBS1PR1S1PR4S1PR5
SCHEMBL5425206 0.80 MAPK14 (0.46) THRATHRBS1PR1S1PR4S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996565-A2 SUBSTITUTED AMINOTHIAZOLE DERIVATIVES WITH ANTI-HCV ACTIVITY Achillion Pharmaceuticals, Inc. (US) 2008-12-03 EP claimed
WO-2007103550-A2 SUBSTITUTED AMINOTHIAZOLE DERIVATIVES WITH ANTI-HCV ACTIVITY ACHILLION PHARMACEUTICALS, INC. (US) 2007-09-13 WO claimed