SCHEMBL4723079

SCHEMBL4723079

CCCNc1cc(-c2cccc(OC)c2)nn(-c2cc(N3CCOCC3)ccc2Cl)c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
MAPT P10636 3/20 0.43
MAPK1 P28482 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
LMNA P02545 1/20 0.43
PKM P14618 1/20 0.43
CYP1A2 P05177 2/20 0.43
CYP1A1 P04798 1/20 0.43
CYP1B1 Q16678 1/20 0.43
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
GSK3B P49841 1/20 0.40
GAK O14976 1/20 0.39
PRKDC P78527 1/20 0.39
ADRA1D P25100 3/20 0.39
ADRA1A P35348 3/20 0.39
ADRA1B P35368 3/20 0.39
HSD17B10 Q99714 2/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4723258 0.92 HTT (0.42) MEN1KMT2AMAPTMAPK1TDP1
SCHEMBL4724315 0.91 MEN1 (0.45) MEN1KMT2AMAPTMAPK1TDP1
SCHEMBL4723995 0.91 GAA (0.50) MEN1KMT2AMAPTMAPK1TDP1
SCHEMBL4722685 0.88 MEN1 (0.46) MEN1KMT2AMAPTMAPK1TDP1
SCHEMBL4723860 0.88 ADRA1D (0.42) MEN1KMT2AMAPTMAPK1TDP1
SCHEMBL4723078 0.83 CYP1A2 (0.41) MEN1KMT2AMAPTMAPK1LMNA
SCHEMBL4724040 0.83 CYP1A2 (0.44) MEN1KMT2AMAPTMAPK1CYP1A2
SCHEMBL4722912 0.82 MAPT (0.49) MEN1KMT2AMAPTMAPK1TDP1
SCHEMBL4722409 0.81 MAPT (0.53) MEN1KMT2AMAPTMAPK1TDP1
SCHEMBL4719751 0.79 ADRA1D (0.44) MEN1KMT2AMAPTTDP1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed