SCHEMBL4723724

SCHEMBL4723724

COc1cc(OC)cc(-c2nn(-c3cc(C(=O)N(C)C)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 3/20 0.42
CYP2D6 P10635 2/20 0.42
CYP1A2 P05177 2/20 0.42
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
RORC P51449 2/20 0.34
F10 P00742 4/20 0.34
ALDH1A1 P00352 1/20 0.34
NTRK1 P04629 2/20 0.34
ALPL P05186 1/20 0.33
ALPI P09923 1/20 0.33
RARG P13631 1/20 0.33
PPARG P37231 1/20 0.33
UGCG Q16739 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
CYP2C9 P11712 2/20 0.33
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722664 0.91 PDE4A (0.41) GRIA2CYP2D6CYP1A2PDE4APDE4B
SCHEMBL4722532 0.90 NOTUM (0.39) CYP2D6CYP1A2PDE4APDE4BPDE4C
SCHEMBL4764994 0.90 PDE4A (0.40) GRIA2CYP2D6CYP1A2PDE4APDE4B
SCHEMBL4718847 0.89 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DNTRK1
SCHEMBL4721150 0.87 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DF10
SCHEMBL4721033 0.86 F10 (0.39) PDE4APDE4BPDE4CPDE4DF10
SCHEMBL4720453 0.86 F10 (0.43) GRIA2CYP2D6CYP1A2PDE4APDE4B
SCHEMBL4720223 0.85 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DALPL
SCHEMBL4719764 0.85 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL4723271 0.84 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed