SCHEMBL4764994

SCHEMBL4764994

COc1cc(OC)cc(-c2nn(-c3cc(C(N)=O)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.40
PDE4B Q07343 2/20 0.40
PDE4C Q08493 2/20 0.40
PDE4D Q08499 2/20 0.40
AR P10275 1/20 0.36
GHSR Q92847 2/20 0.34
NPC1 O15118 2/20 0.34
CSNK1E P49674 1/20 0.34
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
ALPL P05186 1/20 0.33
ALPI P09923 1/20 0.33
CYP2C9 P11712 1/20 0.33
KIF11 P52732 1/20 0.33
UGCG Q16739 1/20 0.33
NTRK1 P04629 1/20 0.33
RORC P51449 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
RIPK2 O43353 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722664 0.92 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DALPL
SCHEMBL4722532 0.91 NOTUM (0.39) PDE4APDE4BPDE4CPDE4DALPL
SCHEMBL4723724 0.90 GRIA2 (0.42) PDE4APDE4BPDE4CPDE4DALPL
SCHEMBL4718847 0.89 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DKIF11
SCHEMBL4721150 0.88 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL4723271 0.87 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DALPL
SCHEMBL4719764 0.86 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DALPL
SCHEMBL4720223 0.86 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DALPL
SCHEMBL4719190 0.85 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DALPL
SCHEMBL4724138 0.85 PDE4A (0.39) PDE4APDE4BPDE4CPDE4DSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed