SCHEMBL4724221

SCHEMBL4724221

CCNc1cc(-c2cc(C)cc(-c3cnco3)c2)nn(-c2cc(NCCO)ccc2C(F)(F)F)c1=O

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.33
PTK2 Q05397 1/20 0.33
IMPDH2 P12268 2/20 0.32
IMPDH1 P20839 1/20 0.32
QPCT Q16769 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722031 0.95 PTK2 (0.33) PTK2IMPDH2IMPDH1
SCHEMBL4724073 0.91 NTRK1 (0.32) NTRK1PTK2IMPDH2IMPDH1QPCT
SCHEMBL4723056 0.90 LMNA (0.32) PTK2IMPDH2IMPDH1
SCHEMBL4718834 0.88 CYP3A4 (0.34)
SCHEMBL4721397 0.88 S1PR1 (0.31)
SCHEMBL4721894 0.86 PTK2 (0.30) PTK2
SCHEMBL4722748 0.86
SCHEMBL4719336 0.85
SCHEMBL4720065 0.85 POLB (0.31)
SCHEMBL4720181 0.85 NTRK1 (0.32) NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed