SCHEMBL4724637

SCHEMBL4724637

CCCOc1ccn[c]c1-c1cccc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 10/20 0.43
HTR1D P28221 3/20 0.43
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
TLR8 Q9NR97 1/20 0.41
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
TSHR P16473 1/20 0.39
PDE5A O76074 2/20 0.38
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
MCHR1 Q99705 1/20 0.38
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4721628 0.94 HTR1B (0.47) HTR1BHTR1DCNR1CNR2TLR8
SCHEMBL4724855 0.89 ENPP1 (0.44) HTR1BHTR1DTLR8MEN1KMT2A
SCHEMBL4724144 0.82 ALDH1A1 (0.41) CNR2MEN1KMT2ATSHRNPC1
SCHEMBL4719990 0.81 CNR1 (0.41) HTR1BHTR1DCNR1CNR2TLR8
SCHEMBL4723779 0.77 TLR8 (0.40) TLR8MEN1KMT2ATSHRPDE5A
SCHEMBL4722971 0.76 CNR1 (0.44) HTR1BHTR1DCNR1CNR2MEN1
SCHEMBL28075369 0.75 HTR1B (0.54) HTR1BHTR1DCNR1CNR2SLC6A4
SCHEMBL4724769 0.75 CNR1 (0.43) HTR1BHTR1DCNR1CNR2MEN1
SCHEMBL4723799 0.74 HTR1B (0.43) HTR1BHTR1DCNR1CNR2TLR8
SCHEMBL4723379 0.74 ALDH1A1 (0.40) HTR1BHTR1DCNR1CNR2TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957495-A1 FUSED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2008-08-20 EP disclosed
WO-2007064045-A1 FUSED HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-06-07 WO disclosed