SCHEMBL4725258

SCHEMBL4725258

COc1cc2ncnc(-c3ccccc3)c2cc1OCc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.57
IRAK1 P51617 1/20 0.56
IRAK4 Q9NWZ3 1/20 0.56
EGFR P00533 8/20 0.56
KDM4E B2RXH2 1/20 0.56
LMNA P02545 1/20 0.56
HPGD P15428 1/20 0.56
HTT P42858 1/20 0.56
KIT P10721 3/20 0.55
LCK P06239 1/20 0.55
MAPK1 P28482 1/20 0.54
WHR1 P49842 1/20 0.52
PDPK1 O15530 1/20 0.52
ACHE P22303 1/20 0.50
BACE1 P56817 1/20 0.50
RET P07949 1/20 0.50
KDR P35968 1/20 0.50
ATM Q13315 1/20 0.50
ELANE P08246 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26102836 0.92 KDM1A (0.53) KDM1AIRAK1IRAK4EGFRKDM4E
SCHEMBL26098937 0.92 KIT (0.56) KDM1AIRAK1IRAK4EGFRKDM4E
SCHEMBL4782102 0.90 WHR1 (0.61) EGFRKDM4ELMNAHPGDHTT
SCHEMBL26101213 0.87 ABCG2 (0.53) KDM1AIRAK1IRAK4EGFRKDM4E
SCHEMBL26099045 0.84 PDGFRB (0.51) KDM1AIRAK1IRAK4EGFRKDM4E
SCHEMBL10296331 0.84 IRAK1 (0.68) KDM1AIRAK1IRAK4EGFRKDM4E
SCHEMBL16281244 0.84 KDM1A (0.60) KDM1AIRAK1IRAK4EGFRKDM4E
SCHEMBL8499854 0.83 EGFR (0.52) KDM1AIRAK1IRAK4EGFRKDM4E
SCHEMBL14417895 0.83 KDM1A (0.58) KDM1AIRAK1IRAK4EGFRKDM4E
SCHEMBL295891 0.83 ENPP1 (0.68) KDM1AIRAK1IRAK4EGFRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008020302-A2 HETEROAROMATIC QUINOLINE-BASED COMPOUNDS AS PHOSPHODIESTERASE (PDE) INHIBITORS PFIZER PRODUCTS INC. (US) 2008-02-21 WO disclosed