SCHEMBL4725523

SCHEMBL4725523

c1ccc2nc(COc3ccc4ncnc(-c5ccncc5)c4c3)ccc2c1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 13/20 0.56
CYP1A2 P05177 2/20 0.55
LGALS3 P17931 1/20 0.55
PDE4D Q08499 1/20 0.55
CYSLTR2 Q9NS75 1/20 0.50
CYSLTR1 Q9Y271 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4725039 0.92 CYSLTR1 (0.57) PDE10ACYP1A2CYSLTR2CYSLTR1
SCHEMBL4783734 0.91 PDE10A (0.59) PDE10ACYP1A2LGALS3PDE4DCYSLTR2
SCHEMBL4730048 0.89 PDE10A (0.44) PDE10ACYP1A2LGALS3PDE4DCYSLTR2
SCHEMBL4728459 0.88 PDE10A (0.56) PDE10ACYP1A2CYSLTR2CYSLTR1
SCHEMBL4725624 0.83 PDE10A (0.60) PDE10ACYP1A2CYSLTR2CYSLTR1
SCHEMBL4726967 0.82 PDE10A (0.52) PDE10ACYP1A2LGALS3PDE4D
SCHEMBL4726394 0.82 PDE10A (0.52) PDE10ACYP1A2LGALS3PDE4D
SCHEMBL4725570 0.81 IP6K1 (0.50)
SCHEMBL4727365 0.81 PIK3CD (0.51) PDE10ACYP1A2CYSLTR2CYSLTR1
SCHEMBL4780024 0.80 CYSLTR1 (0.51) PDE10ACYP1A2CYSLTR2CYSLTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008020302-A2 HETEROAROMATIC QUINOLINE-BASED COMPOUNDS AS PHOSPHODIESTERASE (PDE) INHIBITORS PFIZER PRODUCTS INC. (US) 2008-02-21 WO claimed