SCHEMBL4726154

SCHEMBL4726154

O=C(O)NCCOCc1csc(NC(=O)NCc2ccc(Cl)c(Cl)c2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 11/20 0.42
ROCK2 O75116 10/20 0.42
TRPV1 Q8NER1 3/20 0.42
MAPK1 P28482 2/20 0.41
AURKA O14965 1/20 0.41
DYRK3 O43781 1/20 0.41
PRKD3 O94806 1/20 0.41
PRKCG P05129 1/20 0.41
PRKACA P17612 1/20 0.41
RPS6KB1 P23443 1/20 0.41
MARK3 P27448 1/20 0.41
AKT1 P31749 1/20 0.41
CSNK1D P48730 1/20 0.41
CLK2 P49760 1/20 0.41
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
RPS6KA3 P51812 1/20 0.41
PRKX P51817 1/20 0.41
LIMK1 P53667 1/20 0.41
CSNK2A1 P68400 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4778605 0.91 ROCK1 (0.42) ROCK1ROCK2TRPV1MAPK1AURKA
SCHEMBL4726089 0.91 TSHR (0.50) ROCK1ROCK2TRPV1MAPK1AURKA
SCHEMBL4726401 0.90 LMNA (0.42) ROCK1ROCK2TRPV1MAPK1AURKA
SCHEMBL4725694 0.89 ROCK1 (0.44) ROCK1ROCK2TRPV1MAPK1AURKA
SCHEMBL4778546 0.88 ROCK1 (0.44) ROCK1ROCK2TRPV1MAPK1AURKA
SCHEMBL4780515 0.87 TSHR (0.41) ROCK1ROCK2TRPV1MAPK1AURKA
Hydrochloric Acid SCHEMBL4779977 0.87 ROCK1 (0.43) ROCK1ROCK2TRPV1MAPK1AURKA
SCHEMBL4780046 0.87 TSHR (0.46) ROCK1ROCK2TRPV1MAPK1AURKA
SCHEMBL4777271 0.87 ROCK1 (0.48) ROCK1ROCK2TRPV1MAPK1AURKA
SCHEMBL4777329 0.87 ROCK1 (0.43) ROCK1ROCK2TRPV1MAPK1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008011191-A1 ANTIBACTERIAL HETEROCYCLIC UREAS REPLIDYNE, INC. (US) 2008-01-24 WO claimed
WO-2008011191-A1 ANTIBACTERIAL HETEROCYCLIC UREAS REPLIDYNE, INC. (US) 2008-01-24 WO disclosed