SCHEMBL4728065

SCHEMBL4728065

CC(C)(C)[Si](C)(C)OCCc1cccc(-c2cnc(N)c(C(=O)O)n2)c1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ATR Q13535 13/20 0.44
PRKDC P78527 3/20 0.43
PIK3CD O00329 3/20 0.43
PIK3CA P42336 3/20 0.43
PIK3CG P48736 3/20 0.43
LDHA P00338 1/20 0.43
LDHB P07195 1/20 0.43
ATM Q13315 1/20 0.41
TYRO3 Q06418 1/20 0.40
PIK3CB P42338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4730225 0.81 ATR (0.46) ATRPRKDCPIK3CDPIK3CAPIK3CG
SCHEMBL1166941 0.77 HCRTR2 (0.42)
SCHEMBL4741394 0.75 FOLH1 (0.46)
SCHEMBL11906697 0.73 ATR (0.72) ATRPRKDCPIK3CDPIK3CAPIK3CG
SCHEMBL408691 0.73 GSK3B (0.61) ATRPRKDC
SCHEMBL13401182 0.73 ATR (0.45) ATRPRKDCPIK3CDPIK3CAPIK3CG
SCHEMBL4731377 0.72 ATR (0.40) ATRPRKDCPIK3CDPIK3CAPIK3CG
SCHEMBL16836772 0.72 PTGER4 (0.48)
SCHEMBL318797 0.71 ATR (0.68) ATRPRKDCATM
SCHEMBL3983850 0.71 ATR (0.72) ATRPRKDCPIK3CDPIK3CAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008038010-A1 PYRAZINE DERIVATIVES AND THEIR USE IN THERAPY VERNALIS (R & D) LIMITED (GB) 2008-04-03 WO disclosed