SCHEMBL4728102

SCHEMBL4728102

O=C(N1Cc2ccc(CCCCCl)cc2C1)C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.45
ESR2 Q92731 4/20 0.45
NAMPT P43490 6/20 0.45
ABHD6 Q9BV23 6/20 0.40
S1PR1 P21453 1/20 0.39
MGLL Q99685 1/20 0.39
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
FAAH O00519 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4730749 0.82 NOTUM (0.47) NAMPTS1PR1
SCHEMBL25200985 0.80 ESR1 (0.51) ESR1ESR2ABHD6MGLLHDAC8
SCHEMBL565064 0.77 ESR1 (0.58) ESR1ESR2ABHD6S1PR1HDAC8
SCHEMBL1367276 0.75 ESR1 (0.52) ESR1ESR2ABHD6HDAC8HDAC6
SCHEMBL25199618 0.74 ESR1 (0.57) ESR1ESR2NAMPTABHD6HDAC8
SCHEMBL30412058 0.74 ESR1 (0.57) ESR1ESR2NAMPTABHD6HDAC8
SCHEMBL1366031 0.74 ESR1 (0.48) ESR1ESR2NAMPTABHD6MGLL
SCHEMBL25604135 0.72 ESR2 (0.77) ESR1ESR2ABHD6HDAC8HDAC6
SCHEMBL13439632 0.72 KCNJ1 (0.48) ESR1ESR2NAMPTABHD6MGLL
SCHEMBL5913288 0.71 ESR1 (0.54) ESR1ESR2NAMPTABHD6MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008020306-A2 ISOINDOLE DERIVATIVES PFIZER PRODUCTS INC. (US) 2008-02-21 WO disclosed
WO-2008020306-A2 ISOINDOLE DERIVATIVES PFIZER PRODUCTS INC. (US) 2008-02-21 WO disclosed