SCHEMBL4729062

SCHEMBL4729062

CC(=O)Oc1cc(Cl)cc(OCCC2(C#N)CCN(c3nc4ccc(C(F)(F)F)cc4s3)CC2)c1

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 20/20 0.60
PPARG P37231 14/20 0.60
PPARA Q07869 6/20 0.60
CYP2C9 P11712 4/20 0.58
CYP3A4 P08684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL334892 0.87 PPARD (0.78) PPARDPPARGPPARACYP2C9CYP3A4
SCHEMBL334111 0.79 PPARD (0.47) PPARDPPARGPPARACYP2C9
SCHEMBL10221459 0.79 PPARD (0.65) PPARDPPARGPPARACYP2C9CYP3A4
SCHEMBL10271422 0.77 PPARD (0.81) PPARDPPARGPPARACYP2C9
SCHEMBL334494 0.77 PPARD (0.44) PPARDPPARGPPARACYP2C9CYP3A4
SCHEMBL10221075 0.75 PPARD (1.00) PPARDPPARGPPARACYP2C9CYP3A4
SCHEMBL10221152 0.75 PPARD (0.74) PPARDPPARGPPARACYP2C9
SCHEMBL334583 0.75 PPARD (0.71) PPARDPPARGPPARACYP2C9
SCHEMBL10221097 0.74 PPARD (0.99) PPARDPPARGPPARACYP2C9CYP3A4
SCHEMBL334495 0.73 PPARD (0.41) PPARDPPARGPPARACYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1939189-A1 DERIVATIVE HAVING PPAR AGONISTIC ACTIVITY SHIONOGI & CO., LTD. (JP) 2008-07-02 EP disclosed