SCHEMBL4730504

SCHEMBL4730504

CCC(CC)c1ccc(N(Cc2cccc(-c3ccc(COc4cncc(C(=O)OC)c4)cc3)c2)C(C)C)cc1

nearest known ligand 0.65

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.65
SIRT2 Q8IXJ6 9/20 0.41
SIRT1 Q96EB6 8/20 0.41
SIRT3 Q9NTG7 8/20 0.41
ADAMTS4 O75173 1/20 0.39
MMP13 P45452 1/20 0.39
SMPD1 P17405 1/20 0.37
PSMB5 P28074 2/20 0.37
PTGES O14684 1/20 0.37
ALOX5 P09917 1/20 0.37
LTC4S Q16873 1/20 0.37
FFAR1 O14842 3/20 0.37
GNA15 P30679 1/20 0.37
GRM5 P41594 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4730123 0.92 PTPN1 (0.66) PTPN1SIRT2SIRT1SIRT3PSMB5
SCHEMBL4726653 0.88 PTPN1 (0.60) PTPN1SIRT2SIRT1SIRT3PTGES
SCHEMBL14260784 0.83 PTPN1 (0.56) PTPN1SIRT2SIRT1SIRT3PTGES
SCHEMBL4730748 0.83 PTPN1 (0.45) PTPN1SIRT2SIRT1SIRT3MMP13
SCHEMBL14261277 0.83 PTPN1 (0.54) PTPN1SIRT2SIRT1ADAMTS4PTGES
SCHEMBL14261224 0.82 PTPN1 (0.76) PTPN1ADAMTS4MMP13PTGESALOX5
SCHEMBL14261225 0.82 PTPN1 (0.76) PTPN1ADAMTS4MMP13PTGESALOX5
SCHEMBL14260788 0.82 PTPN1 (0.53) PTPN1SIRT2SIRT1ADAMTS4SMPD1
SCHEMBL6000633 0.82 PTPN1 (0.43) PTPN1SIRT2SIRT1SIRT3MMP13
SCHEMBL14260886 0.81 PTPN1 (0.76) PTPN1PTGESALOX5FFAR1GNA15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033455-A2 BIPHENYL AND HETEROARYL PHENYL DERIVATIVES AS PROTEIN TYROSINE PHOSPHATASES INHIBITORS THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2008-03-20 WO disclosed
WO-2008033455-A2 BIPHENYL AND HETEROARYL PHENYL DERIVATIVES AS PROTEIN TYROSINE PHOSPHATASES INHIBITORS THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2008-03-20 WO disclosed