SCHEMBL4733798

SCHEMBL4733798

CCC(C)(C)C(=O)Nc1cc(CN(C)Cc2ccccc2)c(Br)cn1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 6/20 0.45
CNR1 P21554 3/20 0.45
RIPK1 Q13546 5/20 0.43
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
HDAC1 Q13547 1/20 0.38
CCR5 P51681 1/20 0.37
TMEM97 Q5BJF2 1/20 0.36
SIGMAR1 Q99720 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4783553 0.88 CNR2 (0.53) CNR2CNR1RIPK1NPC1RAB9A
SCHEMBL14206962 0.81 CNR2 (0.45) CNR2CNR1RIPK1
SCHEMBL14206639 0.80 CNR2 (0.59) CNR2CNR1RIPK1ALDH1A1
SCHEMBL4733593 0.79 CNR2 (0.52) CNR2CNR1RIPK1NPC1RAB9A
SCHEMBL4731510 0.78 CNR2 (0.55) CNR2CNR1RIPK1NPC1RAB9A
SCHEMBL14206637 0.77 CNR2 (0.54) CNR2CNR1RIPK1L3MBTL1ALDH1A1
SCHEMBL4732572 0.77 CNR2 (0.46) CNR2CNR1RIPK1NPC1RAB9A
SCHEMBL14206662 0.76 CNR2 (0.56) CNR2CNR1RIPK1
SCHEMBL4734267 0.76 CNR2 (0.50) CNR2CNR1RIPK1NPC1RAB9A
SCHEMBL4730027 0.75 CNR2 (0.42) CNR2CNR1RAB9AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008063625-A2 PYRIDINE COMPOUNDS AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2008-05-29 WO disclosed
WO-2008063625-A2 PYRIDINE COMPOUNDS AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2008-05-29 WO disclosed