SCHEMBL4734015

SCHEMBL4734015

CCC(C)(C)C(=O)Nc1cc(C)cc(C)n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.57
MAPK1 P28482 2/20 0.51
LCK P06239 1/20 0.50
CHRNB2 P17787 1/20 0.49
CHRNB4 P30926 1/20 0.49
CHRNA3 P32297 1/20 0.49
CHRNA4 P43681 1/20 0.49
ALDH1A1 P00352 2/20 0.48
TP53 P04637 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 1/20 0.47
GBA1 P04062 1/20 0.47
RAB9A P51151 1/20 0.47
LMNA P02545 2/20 0.46
MAPT P10636 1/20 0.46
HTT P42858 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
NOS3 P29474 1/20 0.44
NOS2 P35228 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12189258 0.83 LCK (0.55) MAPK1LCKCHRNB2CHRNB4CHRNA3
SCHEMBL14207101 0.82 CNR2 (0.45) CNR2MAPK1LCKCHRNB2CHRNB4
SCHEMBL12182431 0.77 MAPK1 (0.65) MAPK1LCKCHRNB2CHRNB4CHRNA3
SCHEMBL4783898 0.76 CNR2 (0.46) CNR2ALDH1A1NPC1RAB9ALMNA
SCHEMBL30711612 0.76 LCK (0.67) MAPK1LCKCHRNB2CHRNB4CHRNA3
SCHEMBL4504096 0.76 LCK (0.67) MAPK1LCKCHRNB2CHRNB4CHRNA3
SCHEMBL4733265 0.75 CNR2 (0.46) CNR2ALDH1A1NPC1RAB9ALMNA
SCHEMBL14206939 0.75 CNR2 (0.46) CNR2ALDH1A1NPC1RAB9ALMNA
SCHEMBL50044 0.74 LCK (0.60) MAPK1LCKCHRNB2CHRNB4CHRNA3
SCHEMBL9665242 0.74 MAPK1 (0.70) MAPK1LCKCHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008063625-A2 PYRIDINE COMPOUNDS AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2008-05-29 WO disclosed
WO-2008063625-A2 PYRIDINE COMPOUNDS AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2008-05-29 WO disclosed