Austricin

Austricin

SCHEMBL4735162

CC1=CC(=O)C2=C(C)C[C@H](O)[C@@H]3[C@H](OC(=O)[C@H]3C)[C@@H]12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.97
MAPK1 P28482 1/20 0.97
LMNA P02545 1/20 0.97
ALDH1A1 P00352 3/20 0.57
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
CYP19A1 P11511 2/20 0.41
CYP3A4 P08684 1/20 0.36
TAS2R31 P59538 2/20 0.32
TAS2R46 P59540 2/20 0.32
TAS2R10 Q9NYW0 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Austricin SCHEMBL14190527 1.00 CYP1A2 (0.97) CYP1A2MAPK1LMNAALDH1A1MEN1
Austricin SCHEMBL14029373 1.00 CYP1A2 (0.97) CYP1A2MAPK1LMNAALDH1A1MEN1
SCHEMBL8898751 0.85 CYP1A2 (0.72) CYP1A2MAPK1LMNAALDH1A1MEN1
SCHEMBL14215974 0.85 CYP1A2 (0.72) CYP1A2MAPK1LMNAALDH1A1MEN1
8Alpha-Acetoxyachillin SCHEMBL8959436 0.81 ALDH1A1 (0.70) CYP1A2MAPK1LMNAALDH1A1MEN1
SCHEMBL3031437 0.73 ALDH1A1 (1.00) CYP1A2MAPK1LMNAALDH1A1MEN1
Desacetoxymatricarin SCHEMBL14190533 0.73 CYP1A2 (1.00) CYP1A2MAPK1LMNAALDH1A1MEN1
Desacetoxymatricarin SCHEMBL5004433 0.73 CYP1A2 (1.00) CYP1A2MAPK1LMNAALDH1A1MEN1
Desacetoxymatricarin SCHEMBL14029298 0.73 CYP1A2 (1.00) CYP1A2MAPK1LMNAALDH1A1MEN1
Desacetoxymatricarin SCHEMBL3458919 0.73 CYP1A2 (1.00) CYP1A2MAPK1LMNAALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4040154-B1 IMMUNOCHROMATOGRAPHY FUJIFILM CORP (JP) 2025-06-25 EP claimed
EP-4040155-B1 IMMUNOCHROMATOGRAPHY FUJIFILM CORP (JP) 2024-11-27 EP claimed
WO-2024181633-A1 COMPOSITION FOR PREVENTING, AMELIORATING, OR TREATING STRIAE DISTENSAE COMPRISING EXTRACT OF CORCHORUS OLITORIUS L. AND COMPLEX EXTRACT OF TARAXACUM PLATYCARPUM AND HORDEUM VULGARE L. 주식회사 바이오코스 2024-09-06 WO disclosed
US-20200188464-A1 COMPOSITION FOR PROTECTING LIVER COMPRISING DANDELION EXTRACT AND LEMON BALM EXTRACT PHYTONUTRIMEDI CO., LTD. (KR) 2020-06-18 US disclosed
EP-3653220-A2 COMPOSITION FOR PROTECTING LIVER COMPRISING DANDELION EXTRACT AND LEMON BALM EXTRACT Phytonutrimedi Co., Ltd. (KR) 2020-05-20 EP disclosed
WO-2018056746-A1 SWEET-TASTING PROTEIN BRAZZEIN VARIANT HAVING ANTIALLERGIC ACTIVITY 주식회사 바이오스위트 2018-03-29 WO disclosed
US-20080145465-A1 Sesquiterpene lactone extract from artemisia leucodes for reducing inflammation and down-regulating pro-inflammatory gene expression RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2008-06-19 US disclosed
WO-2008054756-A2 SESQUITERPENE LACTONES FROM ARTEMISIA LEUCODES AS ANTI-INFLAMMATORY AND GENE REGULATORS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2008-05-08 WO disclosed
US-5663196-A ADMINISTERING A SESQUITERPENE LACTONE TO AN ANIMAL BOSTON UNIVERSITY (US) 1997-09-02 US disclosed
WO-1995006476-A1 METHODS AND COMPOSITIONS FOR TREATING NEOPLASTIC DISORDERS TRUSTEES OF BOSTON UNIVERSITY (US) 1995-03-09 WO disclosed