SCHEMBL4737052

SCHEMBL4737052

Cc1nc(C(C)C)c(Sc2cc(Cl)cc(Cl)c2)n1Cc1ccncc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.39
TDP1 Q9NUW8 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
BRD4 O60885 1/20 0.34
IDO1 P14902 1/20 0.33
SOS1 Q07889 1/20 0.33
HSP90B1 P14625 1/20 0.33
TRAP1 Q12931 1/20 0.33
PDE10A Q9Y233 1/20 0.33
GALR3 O60755 1/20 0.33
NR2F2 P24468 1/20 0.33
RAB9A P51151 1/20 0.33
TYMS P04818 1/20 0.32
HTT P42858 1/20 0.32
KDM4E B2RXH2 1/20 0.32
TLR9 Q9NR96 1/20 0.31
TLR8 Q9NR97 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
P2RX3 P56373 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1075136 0.87 KCNH2 (0.36) KCNH2TDP1MEN1KMT2AIDO1
SCHEMBL14439807 0.86 KCNH2 (0.38) KCNH2TDP1MEN1KMT2AIDO1
SCHEMBL5852651 0.85 KCNH2 (0.35) KCNH2TDP1MEN1KMT2AIDO1
SCHEMBL6957548 0.85 KCNH2 (0.35) KCNH2TDP1MEN1KMT2AIDO1
SCHEMBL14439809 0.85 KCNH2 (0.35) KCNH2TDP1MEN1KMT2AIDO1
SCHEMBL8343685 0.85 KCNH2 (0.37) KCNH2TDP1MEN1KMT2AIDO1
SCHEMBL6967722 0.84 TDP1 (0.34) KCNH2TDP1MEN1KMT2AIDO1
SCHEMBL6973648 0.83 KCNH2 (0.34) KCNH2TDP1HSP90B1TRAP1
SCHEMBL7077305 0.83 KCNH2 (0.34) KCNH2TDP1HSP90B1TRAP1
SCHEMBL7084120 0.83 KCNH2 (0.34) KCNH2TDP1MEN1KMT2AHSP90B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720856-B1 HIV INTEGRASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2013-08-14 EP claimed
EP-1569931-B1 HETEROCYCLIC COMPOUNDS AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2008-10-08 EP claimed
EP-1569933-B1 PYRROLIDINE AND AZETIDINE COMPOUNDS AS CCR5 ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2008-07-23 EP claimed
EP-1172097-B1 PROCESS FOR PRODUCING MEDICINAL COMPOSITION OF A BASIC HYDROPHOBIC MEDICINAL COMPOUND SHIONOGI & CO (JP) 2004-09-08 EP claimed