SCHEMBL4737083

SCHEMBL4737083

O=C(O)c1cnc2[nH]ncc2c1N1CCOC(CO)C1

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 7/20 0.64
CHEK2 O96017 4/20 0.64
PDE10A Q9Y233 1/20 0.42
HDAC6 Q9UBN7 1/20 0.39
PDE4B Q07343 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LRRK2 Q5S007 1/20 0.37
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
SYK P43405 3/20 0.36
ABL1 P00519 1/20 0.36
JAK3 P52333 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4737061 0.90 CHEK1 (0.65) CHEK1CHEK2PDE10APDE4BALDH1A1
SCHEMBL4737214 0.89 CHEK1 (0.59) CHEK1CHEK2PDE10APDE4BALDH1A1
SCHEMBL4738311 0.89 CHEK1 (0.64) CHEK1CHEK2PDE10APDE4BALDH1A1
SCHEMBL14163041 0.86 CHEK1 (0.86) CHEK1CHEK2PDE10APDE4BADORA1
SCHEMBL14162805 0.86 CHEK1 (0.86) CHEK1CHEK2PDE10APDE4BADORA1
SCHEMBL4735382 0.83 CHEK1 (0.58) CHEK1CHEK2PDE10APDE4BALDH1A1
SCHEMBL4738914 0.80 CHEK1 (0.63) CHEK1CHEK2PDE10AHDAC6PDE4B
SCHEMBL4738683 0.79 CHEK1 (0.75) CHEK1CHEK2HDAC6PDE4BALDH1A1
SCHEMBL14162782 0.79 CHEK1 (0.70) CHEK1CHEK2PDE4BALDH1A1JAK3
SCHEMBL14162773 0.79 CHEK1 (0.67) CHEK1CHEK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008075007-A1 MORPHOLINO-SUBSTITUTED BICYCLOHETEROARYL COMPOUNDS AND THEIR USE AS ANTI CANCER AGENTS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2008-06-26 WO disclosed