SCHEMBL4738683

SCHEMBL4738683

CCNC(=O)c1cnc2[nH]ncc2c1N1CCOC(CN)C1

nearest known ligand 0.75

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 13/20 0.75
CHEK2 O96017 9/20 0.75
PDE4B Q07343 1/20 0.38
JAK3 P52333 2/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
TYK2 P29597 1/20 0.37
PAK1 Q13153 1/20 0.35
ALDH1A1 P00352 1/20 0.35
AKT2 P31751 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4738914 0.89 CHEK1 (0.63) CHEK1CHEK2PDE4BJAK3JAK2
SCHEMBL14162764 0.86 CHEK1 (0.74) CHEK1CHEK2PDE4BJAK3PAK1
SCHEMBL4803059 0.86 CHEK1 (1.00) CHEK1CHEK2PDE4B
SCHEMBL14162773 0.84 CHEK1 (0.67) CHEK1CHEK2JAK3JAK2JAK1
SCHEMBL14162782 0.83 CHEK1 (0.70) CHEK1CHEK2PDE4BJAK3PAK1
SCHEMBL4737061 0.80 CHEK1 (0.65) CHEK1CHEK2PDE4BJAK3PAK1
SCHEMBL4737083 0.79 CHEK1 (0.64) CHEK1CHEK2PDE4BJAK3ALDH1A1
SCHEMBL14162801 0.79 CHEK1 (0.86) CHEK1CHEK2PDE4B
SCHEMBL4738639 0.79 CHEK1 (1.00) CHEK1CHEK2AKT2
SCHEMBL21067384 0.79 CHEK1 (1.00) CHEK1CHEK2AKT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008075007-A1 MORPHOLINO-SUBSTITUTED BICYCLOHETEROARYL COMPOUNDS AND THEIR USE AS ANTI CANCER AGENTS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2008-06-26 WO disclosed
WO-2008075007-A1 MORPHOLINO-SUBSTITUTED BICYCLOHETEROARYL COMPOUNDS AND THEIR USE AS ANTI CANCER AGENTS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2008-06-26 WO disclosed