SCHEMBL4737413

SCHEMBL4737413

Clc1ncnc2c1-c1ccc(Br)cc1CC2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 4/20 0.46
SRD5A1 P18405 2/20 0.39
SRD5A2 P31213 1/20 0.39
CYP19A1 P11511 6/20 0.38
CYP11B1 P15538 6/20 0.38
CYP11B2 P19099 6/20 0.38
SLC11A2 P49281 1/20 0.38
PARP10 Q53GL7 1/20 0.36
PARP11 Q9NR21 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
GABRG2 P18507 2/20 0.32
GABRB3 P28472 2/20 0.32
GABRA5 P31644 2/20 0.32
GABRA1 P14867 1/20 0.32
GABRA3 P34903 1/20 0.32
GABRA2 P47869 1/20 0.32
PTAFR P25105 1/20 0.32
METAP1 P53582 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4740750 0.82 TYMS (0.46) TYMSSRD5A1SRD5A2CYP19A1CYP11B1
SCHEMBL14148129 0.82 TYMS (0.35) TYMS
SCHEMBL4739932 0.73 EGFR (0.40) TYMSLMNAMAPT
SCHEMBL204100 0.70 SRD5A1 (0.64) TYMSSRD5A1SRD5A2CYP19A1CYP11B1
SCHEMBL31268305 0.70 SRD5A1 (0.64) TYMSSRD5A1SRD5A2CYP19A1CYP11B1
SCHEMBL1869749 0.67 CYP19A1 (0.47) TYMSSRD5A1SRD5A2CYP19A1CYP11B1
SCHEMBL6651001 0.67 TYMS (0.59) TYMSSRD5A1SRD5A2CYP19A1CYP11B1
SCHEMBL4817935 0.66 SRD5A1 (0.60) TYMSSRD5A1SRD5A2CYP19A1CYP11B1
SCHEMBL20229560 0.65 TYMS (0.47) TYMSSRD5A1SRD5A2CYP19A1CYP11B1
SCHEMBL20797143 0.65 SRD5A1 (0.57) TYMSSRD5A1SRD5A2CYP19A1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed