SCHEMBL473901

SCHEMBL473901

CC(c1ccc(-c2ccc(F)cc2)cc1Cl)C(O)(c1ccc(C#N)cc1)C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 8/20 0.47
AR P10275 3/20 0.44
KIF11 P52732 3/20 0.40
PTPN5 P54829 1/20 0.37
PGR P06401 1/20 0.36
PDE2A O00408 1/20 0.36
TNF P01375 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
EGFR P00533 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474038 0.90 HSD11B1 (0.43) HSD11B1ARKIF11PTPN5PDE2A
SCHEMBL473960 0.88 AR (0.41) HSD11B1ARPTPN5
SCHEMBL473964 0.85 HSD11B1 (0.43) HSD11B1ARKIF11TNF
SCHEMBL473894 0.85 HSD11B1 (0.43) HSD11B1ARTNF
SCHEMBL12164142 0.85 HSD11B1 (0.43) HSD11B1ARKIF11TNF
SCHEMBL12164141 0.85 HSD11B1 (0.43) HSD11B1ARTNF
SCHEMBL473998 0.84 AR (0.47) HSD11B1ARKIF11PDE2A
SCHEMBL15520327 0.83 HSD11B1 (0.41) HSD11B1ARKIF11TNFCYP11B1
SCHEMBL15520147 0.82 HSD11B1 (0.41) HSD11B1ARKIF11TNFCYP11B1
SCHEMBL473957 0.81 AR (0.41) HSD11B1ARPTPN5TNFCYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed