SCHEMBL4739665

SCHEMBL4739665

C#CCNc1nc2c(s1)CC(N)CC2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
ROCK2 O75116 3/20 0.37
MAPT P10636 3/20 0.37
TP53 P04637 1/20 0.37
DRD3 P35462 4/20 0.36
DRD2 P14416 3/20 0.36
HRH2 P25021 2/20 0.36
ADRA2A P08913 2/20 0.36
DRD4 P21917 2/20 0.36
ADRB2 P07550 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
HTR1B P28222 1/20 0.36
HTR2A P28223 1/20 0.36
HTR7 P34969 1/20 0.36
ADRA1A P35348 1/20 0.36
HRH1 P35367 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14146290 1.00 NPC1 (0.42) NPC1RAB9ASMN1; SMN2ROCK2MAPT
Hydrochloric Acid SCHEMBL7311991 0.83 ADRA2A (0.43) NPC1RAB9ASMN1; SMN2ROCK2MAPT
Bromide SCHEMBL7317103 0.81 DRD3 (0.48) NPC1RAB9ASMN1; SMN2ROCK2MAPT
SCHEMBL4786177 0.78 DRD3 (0.62) NPC1RAB9ASMN1; SMN2ROCK2DRD3
SCHEMBL14146078 0.78 DRD3 (0.62) NPC1RAB9ASMN1; SMN2ROCK2DRD3
Bromide SCHEMBL7322483 0.78 NPC1 (0.43) NPC1RAB9ASMN1; SMN2ROCK2MAPT
SCHEMBL14146259 0.76 DRD3 (0.47) NPC1RAB9ASMN1; SMN2ROCK2DRD3
Bromide SCHEMBL7319918 0.74 MAPT (0.47) NPC1RAB9AROCK2MAPTTP53
SCHEMBL14146286 0.73 DRD3 (0.35) NPC1RAB9ASMN1; SMN2ROCK2DRD3
SCHEMBL14146258 0.73 DRD3 (0.35) NPC1RAB9ASMN1; SMN2ROCK2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008086353-A1 PROPARGYL-CONTAINING DERIVATIVES OF TETRAHYDRO-BENZTHIAZOLES AND METHODS OF MAKING AND USING THE SAME ZURAWSKI VINCENT R JR (US) 2008-07-17 WO disclosed
WO-2008086353-A1 PROPARGYL-CONTAINING DERIVATIVES OF TETRAHYDRO-BENZTHIAZOLES AND METHODS OF MAKING AND USING THE SAME ZURAWSKI VINCENT R JR (US) 2008-07-17 WO disclosed