SCHEMBL4739906

SCHEMBL4739906

Nc1nc2c(c(Nc3ccccc3)n1)-c1ccc(Cl)cc1CC2

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TYMS P04818 2/20 0.49
EGFR P00533 5/20 0.45
KDR P35968 2/20 0.43
CDK9 P50750 1/20 0.42
BCL6 P41182 2/20 0.42
CCNA2 P20248 3/20 0.41
CDK2 P24941 3/20 0.41
AGPAT2 O15120 1/20 0.38
ACHE P22303 2/20 0.37
BRAF P15056 1/20 0.37
NR1I2 O75469 1/20 0.37
AHR P35869 1/20 0.37
PLK1 P53350 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739911 0.79 TYMS (0.52) TYMSACHE
SCHEMBL14148121 0.78 TYMS (0.63) TYMS
SCHEMBL8261591 0.78 TYMS (0.59) TYMS
SCHEMBL12391853 0.77 KDR (0.51) EGFRKDRBCL6CCNA2CDK2
SCHEMBL12391875 0.76 EGFR (0.68) EGFRKDRBRAF
SCHEMBL14148437 0.76 TYMS (0.56) TYMSCCNA2CDK2
SCHEMBL12391879 0.76 KDR (0.63) EGFRKDRBCL6CCNA2CDK2
SCHEMBL4787500 0.70 TYMS (0.50) TYMS
SCHEMBL12391871 0.69 KDR (0.51) EGFRKDRACHE
SCHEMBL12391887 0.69 EGFR (0.50) EGFRKDRBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed