SCHEMBL4787500

SCHEMBL4787500

Nc1nc2c(c(-c3ccc(F)cc3)n1)-c1ccc(Cl)cc1CC2

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TYMS P04818 3/20 0.50
ADORA2A P29274 12/20 0.40
ADORA1 P30542 11/20 0.40
DPP4 P27487 1/20 0.39
HSP90AB1 P08238 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
ADORA2B P29275 1/20 0.37
HRH2 P25021 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
PIKFYVE Q9Y2I7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4742391 0.91 TYMS (0.45) TYMSADORA2AADORA1DPP4HSP90AB1
SCHEMBL4739911 0.88 TYMS (0.52) TYMSADORA2AADORA1HSP90AB1ADORA2B
SCHEMBL4740440 0.85 TYMS (0.41) TYMSADORA2AADORA1ADORA3ADORA2B
SCHEMBL4736837 0.79 TYMS (0.38) TYMSADORA2AADORA1ADORA3ADORA2B
SCHEMBL4737447 0.79 TYMS (0.38) TYMSADORA2AADORA1
SCHEMBL4737435 0.79 TYMS (0.47) TYMS
SCHEMBL8261591 0.79 TYMS (0.59) TYMSHSP90AB1
SCHEMBL14148121 0.79 TYMS (0.63) TYMSHSP90AB1
SCHEMBL14148437 0.77 TYMS (0.56) TYMSHSP90AB1
SCHEMBL4737411 0.74 ADORA2A (0.39) TYMSADORA2AADORA1PIKFYVE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed
WO-2008086158-A1 BENZODIHYDROQUINAZOLINE AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-17 WO disclosed