SCHEMBL4740298

SCHEMBL4740298

O=C(c1ccoc1)N(Cc1ccc(C(F)(F)F)nc1)c1ccc(F)cc1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 5/20 0.39
GPBAR1 Q8TDU6 1/20 0.36
LMNA P02545 1/20 0.36
PDK1 Q15118 3/20 0.36
HDAC11 Q96DB2 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
PDK2 Q15119 1/20 0.36
PDK3 Q15120 1/20 0.36
PDK4 Q16654 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
TRPM8 Q7Z2W7 1/20 0.36
CXCR2 P25025 1/20 0.35
NR1H4 Q96RI1 1/20 0.35
BCL2A1 Q16548 1/20 0.34
KCNH2 Q12809 1/20 0.34
CACNA2D1 P54289 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4737132 0.82 MAPK14 (0.44) MAPK14PDK1HDAC11HDAC6HSP90AA1
SCHEMBL4785417 0.81 CACNA1H (0.41) MAPK14LMNAPDK1HSP90AA1HSP90AB1
SCHEMBL4737668 0.81 GAA (0.56) MAPK14PDK1HDAC11HDAC6HDAC8
SCHEMBL4738913 0.78 MAOB (0.40) MAPK14LMNACACNA2D1
SCHEMBL8193274 0.77 MAPK14 (0.42) MAPK14LMNAPDK1HSP90AA1CXCR2
SCHEMBL4734905 0.77 HDAC3 (0.40)
SCHEMBL4737347 0.76 DRD4 (0.43) MAPK14LMNACXCR2
SCHEMBL4735156 0.75 KCNH2 (0.39) MAPK14LMNAPDK1HSP90AA1HSP90AB1
SCHEMBL4735318 0.75 OPRM1 (0.37) MAPK14CXCR2CACNA2D1
SCHEMBL4733936 0.73 OPRM1 (0.49) CACNA2D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed