SCHEMBL4740410

SCHEMBL4740410

O=C(O)CNC(=O)c1c(O)n(Cc2ccccc2Br)c(Cc2ccccc2Cl)nc1=O

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGLN3 Q9H6Z9 8/20 0.47
EGLN1 Q9GZT9 9/20 0.40
TP53 P04637 1/20 0.39
EGLN2 Q96KS0 3/20 0.38
MEN1 O00255 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
KMT2A Q03164 1/20 0.37
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4994580 0.88 EGLN3 (0.49) EGLN3EGLN1TP53EGLN2MEN1
SCHEMBL4738011 0.79 EGLN3 (0.52) EGLN3EGLN1TP53CYP2C19LMNA
SCHEMBL4737678 0.75 EGLN3 (0.48) EGLN3EGLN1TP53EGLN2MEN1
SCHEMBL4992689 0.74 EGLN3 (0.63) EGLN3EGLN1TP53MEN1CYP2C9
SCHEMBL3423804 0.74 EGLN3 (0.69) EGLN3EGLN1TP53EGLN2MEN1
SCHEMBL15419450 0.73 EGLN3 (0.58) EGLN3EGLN1TP53EGLN2MEN1
SCHEMBL1641809 0.72 EGLN3 (0.65) EGLN3EGLN1EGLN2MEN1KMT2A
SCHEMBL4739942 0.72 ALDH1A1 (0.45) MEN1CYP2C9CYP2C19KMT2ALMNA
SCHEMBL12727318 0.72 EGLN3 (0.74) EGLN3EGLN1TP53EGLN2MEN1
SCHEMBL1641768 0.72 EGLN3 (0.74) EGLN3EGLN1TP53EGLN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008089051-A1 N-SUBSTITUTED GLYCINE DERIVATIVES: PROLYL HYDROXYLASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-24 WO claimed