SCHEMBL4740741

SCHEMBL4740741

O=c1[nH]c2c(O)ccc(CCNCc3ccc4[nH]c(CO)nc4c3)c2s1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 17/20 0.56
ABCB11 O95342 2/20 0.47
ADRB1 P08588 5/20 0.45
DRD2 P14416 5/20 0.45
ADRA1D P25100 4/20 0.45
PDE4A P27815 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14099843 0.80 ADRB2 (0.53) ADRB2ABCB11ADRB1DRD2ADRA1D
SCHEMBL4738429 0.76 ADRB2 (0.38) ADRB2
SCHEMBL8879323 0.72 ADRB2 (0.61) ADRB2ABCB11ADRB1DRD2PDE4A
SCHEMBL14104153 0.72 ADRB2 (0.61) ADRB2ABCB11ADRB1DRD2ADRA1D
SCHEMBL9522342 0.72 ADRB2 (0.72) ADRB2ABCB11ADRB1DRD2ADRA1D
SCHEMBL4753827 0.71 ADRB2 (0.55) ADRB2ABCB11ADRB1DRD2ADRA1D
SCHEMBL14100066 0.71 ADRB2 (0.60) ADRB2ABCB11ADRB1DRD2ADRA1D
Hydrochloric Acid SCHEMBL8882013 0.71 ADRB2 (0.71) ADRB2ABCB11ADRB1DRD2ADRA1D
SCHEMBL14077127 0.70 ADRB2 (0.56) ADRB2ABCB11ADRB1DRD2PDE4A
SCHEMBL9520760 0.69 ADRB2 (0.66) ADRB2ABCB11ADRB1DRD2ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008096129-A1 NITROGEN CONTAINING HETROCYCLIC COMPOUNDS USEFUL AS BIFUNCTIONAL MODULATORS OF M3 RECEPTORS AND BETA- 2 RECEPTORS ARGENTA DISCOVERY LTD (GB) 2008-08-14 WO disclosed