SCHEMBL4741007

SCHEMBL4741007

[CH2]c1[nH]c2ccccc2c1C

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 2/20 0.61
ALDH1A1 P00352 6/20 0.50
HSD17B10 Q99714 3/20 0.50
DAO P14920 1/20 0.50
DDO Q99489 1/20 0.50
GPR3 P46089 1/20 0.50
KIF11 P52732 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C19 P33261 1/20 0.45
TNKS2 Q9H2K2 1/20 0.45
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
RAB9A P51151 1/20 0.44
GAA P10253 2/20 0.44
HPGD P15428 2/20 0.44
MAPT P10636 2/20 0.44
RXFP1 Q9HBX9 1/20 0.44
ALOX15 P16050 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3092106 0.84 GAA (0.57) AHRALDH1A1HSD17B10DAODDO
SCHEMBL7195762 0.78 AHR (0.70) AHRALDH1A1HSD17B10DAODDO
SCHEMBL154593 0.76 AHR (1.00) AHRALDH1A1HSD17B10DAODDO
SCHEMBL29420757 0.76 AHR (1.00) AHRALDH1A1HSD17B10DAODDO
Hydrochloric Acid SCHEMBL8462943 0.76 AHR (0.59) AHRALDH1A1HSD17B10DAODDO
SCHEMBL3228514 0.73 ALDH1A1 (0.50) AHRALDH1A1HSD17B10GPR3KIF11
SCHEMBL6817362 0.73 AHR (0.61) AHRALDH1A1HSD17B10DAODDO
SCHEMBL21260226 0.73 AHR (0.61) AHRALDH1A1HSD17B10DAODDO
SCHEMBL7897739 0.73 AHR (0.61) AHRALDH1A1HSD17B10DAODDO
SCHEMBL7495864 0.73 AHR (0.61) AHRALDH1A1HSD17B10DAODDO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6194451-B1 PREVENT RELEASE TUMOR NECROSIS FACTOR; ANTIINFLAMMATORY AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2001-02-27 US claimed
CN-105555763-B indole-carboxamide derivatives 豪夫迈·罗氏有限公司 2018-04-17 CN disclosed
CN-105308024-B The nitrogenous heteroaromatic amide compound of two ring types 安斯泰来制药株式会社 2017-10-27 CN disclosed
CN-105246895-B Piperazino [1, 2-a ] indol-1-ones and [1, 4] diazacyclo [1, 2-a ] indol-1-ones 豪夫迈·罗氏有限公司 2017-09-22 CN disclosed
CN-104540829-B Piperazino[1,2-a]indol-1-ones and [1,4]diazepino[1,2-a]indol-1-one 霍夫曼-拉罗奇有限公司 2017-04-26 CN disclosed
WO-2008104756-A1 UREA DERIVATIVES AND THEIR THERAPEUTIC USE SERENTIS LIMITED (GB) 2008-09-04 WO disclosed
EP-0722436-A4 MERCAPTOSULFIDE METALLOPROTEINASE INHIBITORS UNIV FLORIDA STATE (US) 1996-11-20 EP disclosed
EP-0722436-A1 MERCAPTOSULFIDE METALLOPROTEINASE INHIBITORS FLORIDA STATE UNIVERSITY (US) 1996-07-24 EP disclosed
WO-1995009833-A1 MERCAPTOSULFIDE METALLOPROTEINASE INHIBITORS FLORIDA STATE UNIVERSITY (US) 1995-04-13 WO disclosed