SCHEMBL4741743

SCHEMBL4741743

O=C(Nc1oc(-c2ccccc2)nc1-c1ccccc1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADCY1 Q08828 2/20 0.65
LMNA P02545 2/20 0.56
ALDH1A1 P00352 2/20 0.56
ADCY8 P40145 1/20 0.54
KCNK3 O14649 1/20 0.54
TP53 P04637 1/20 0.51
P2RX1 P51575 1/20 0.50
PTGS1 P23219 2/20 0.49
GAA P10253 1/20 0.49
THRB P10828 1/20 0.48
TRPV1 Q8NER1 1/20 0.48
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4787849 0.88 ADCY1 (0.49) ADCY1TP53PTGS1TRPV1
SCHEMBL4259960 0.84 SMO (0.66) ADCY1LMNAALDH1A1ADCY8KCNK3
SCHEMBL4737638 0.84 KDR (0.55) LMNAALDH1A1GAAMAPT
SCHEMBL14148561 0.83 TP53 (0.50) ADCY1ALDH1A1TP53MAPT
SCHEMBL14148500 0.82 ADORA1 (0.62) LMNAALDH1A1KCNK3MAPT
SCHEMBL7744086 0.80 KDR (0.51) ADCY1ALDH1A1TP53P2RX1
SCHEMBL14148491 0.80 KDM4E (0.66) ADCY1LMNAKCNK3TP53THRB
SCHEMBL7744087 0.79 KDR (0.46) ADCY1LMNAALDH1A1KCNK3TP53
SCHEMBL20598167 0.79 ADCY1 (1.00) ADCY1LMNAALDH1A1ADCY8TP53
SCHEMBL4740831 0.78 SMN1; SMN2 (0.62) ADCY1LMNAALDH1A1ADCY8GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008090382-A1 THIAZOLE AND OXAZOLE DERIVATIVES FOR USE IN THE TREATMENT OF PRION DISEASES, CANCER AND CONDITIONS OF THE CENTRAL NERVOUS SYSTEM AS WELL AS IN THE REGULATION OF STEM CELLS THE UNIVERSITY OF SHEFFIELD (GB) 2008-07-31 WO disclosed