SCHEMBL4743902

SCHEMBL4743902

CC1CN(Cc2ccn(-c3cccnc3N3CCC(Nc4cccc(F)c4)CC3)n2)CC(C)N1

nearest known ligand 0.84

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MLNR O43193 19/20 0.84
CYP3A4 P08684 4/20 0.52
CYP2D6 P10635 3/20 0.52
GHSR Q92847 2/20 0.52
CYP1A2 P05177 1/20 0.52
KDM4E B2RXH2 1/20 0.43
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2010875 1.00 MLNR (0.84) MLNRCYP3A4CYP2D6GHSRCYP1A2
SCHEMBL2004322 0.91 MLNR (1.00) MLNRCYP3A4CYP2D6GHSRCYP1A2
Hydrochloric Acid SCHEMBL2009168 0.90 MLNR (0.98) MLNRCYP3A4CYP2D6GHSRCYP1A2
SCHEMBL2005788 0.85 MLNR (0.78) MLNRCYP3A4CYP2D6GHSRCYP1A2
SCHEMBL4690685 0.84 MLNR (1.00) MLNRCYP3A4CYP2D6GHSRCYP1A2
SCHEMBL2009415 0.84 MLNR (1.00) MLNRCYP3A4CYP2D6GHSRCYP1A2
SCHEMBL2008839 0.83 MLNR (0.85) MLNRCYP3A4CYP2D6GHSRKCNH2
SCHEMBL3134464 0.83 MLNR (0.85) MLNRCYP3A4CYP2D6GHSRCYP1A2
SCHEMBL2011312 0.81 MLNR (0.62) MLNRCYP3A4CYP2D6GHSRCYP1A2
SCHEMBL2007976 0.80 MLNR (1.00) MLNRCYP3A4CYP2D6GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960390-A1 BIARYL COMPOUNDS USEFUL AS AGONISTS OF THE GPR38 RECEPTOR GLAXO GROUP LIMITED (GB) 2008-08-27 EP claimed
WO-2007065669-A1 BIARYL COMPOUNDS USEFUL AS AGONISTS OF THE GPR38 RECEPTOR GLAXO GROUP LIMITED (GB) 2007-06-14 WO claimed