SCHEMBL4690685

SCHEMBL4690685

CC1CN(Cc2ccn(-c3cccnc3N3CCC(Oc4cccc(F)c4)CC3)n2)CC(C)N1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MLNR O43193 13/20 1.00
CYP3A4 P08684 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
GHSR Q92847 1/20 0.36
CHRM4 P08173 3/20 0.36
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
KCNH2 Q12809 2/20 0.34
HRH1 P35367 1/20 0.34
CCR3 P51677 1/20 0.34
SCN9A Q15858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2009415 1.00 MLNR (1.00) MLNRCYP3A4CYP1A2CYP2D6GHSR
SCHEMBL2009345 0.92 MLNR (1.00) MLNR
SCHEMBL2007976 0.91 MLNR (1.00) MLNRCYP3A4CYP2D6GHSRCHRM4
SCHEMBL2012437 0.85 MLNR (1.00) MLNRCYP3A4KCNH2SCN9A
SCHEMBL3134434 0.84 MLNR (0.73) MLNRKCNH2HRH1CCR3SCN9A
SCHEMBL4743902 0.84 MLNR (0.84) MLNRCYP3A4CYP1A2CYP2D6GHSR
SCHEMBL2010875 0.84 MLNR (0.84) MLNRCYP3A4CYP1A2CYP2D6GHSR
SCHEMBL3128327 0.83 MLNR (0.85) MLNRCYP3A4CHRM4
SCHEMBL2010301 0.80 MLNR (0.66) MLNRSLC6A4SLC6A3
SCHEMBL2004322 0.80 MLNR (1.00) MLNRCYP3A4CYP1A2CYP2D6GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960390-A1 BIARYL COMPOUNDS USEFUL AS AGONISTS OF THE GPR38 RECEPTOR GLAXO GROUP LIMITED (GB) 2008-08-27 EP disclosed
WO-2007065669-A1 BIARYL COMPOUNDS USEFUL AS AGONISTS OF THE GPR38 RECEPTOR GLAXO GROUP LIMITED (GB) 2007-06-14 WO disclosed