SCHEMBL4744494

SCHEMBL4744494

CC(C)CNC(=O)CN1CCN(CCCCCOc2ccc3c(-c4ccc(Cl)cc4)coc3c2)CC1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.50
PDK1 Q15118 1/20 0.45
PDK2 Q15119 1/20 0.45
SIGMAR1 Q99720 1/20 0.44
BCHE P06276 2/20 0.43
ACHE P22303 2/20 0.43
ALDH2 P05091 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4742644 0.91 HRH3 (0.52) HRH3PDK1PDK2SIGMAR1BCHE
SCHEMBL4742617 0.90 HRH3 (0.53) HRH3PDK1PDK2SIGMAR1BCHE
SCHEMBL4745561 0.90 HRH3 (0.53) HRH3PDK1PDK2SIGMAR1BCHE
SCHEMBL4744978 0.90 HRH3 (0.54) HRH3PDK1PDK2BCHEACHE
SCHEMBL4741928 0.89 HRH3 (0.54) HRH3PDK1PDK2SIGMAR1BCHE
SCHEMBL4742019 0.89 HRH3 (0.49) HRH3PDK1PDK2SIGMAR1BCHE
SCHEMBL4788438 0.89 HRH3 (0.49) HRH3PDK1PDK2SIGMAR1BCHE
SCHEMBL4744473 0.89 HRH3 (0.50) HRH3PDK1PDK2SIGMAR1
SCHEMBL4744484 0.89 HRH3 (0.47) HRH3PDK1PDK2SIGMAR1BCHE
SCHEMBL4742556 0.88 HRH3 (0.54) HRH3PDK1PDK2SIGMAR1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008107321-A1 HETEROCYCLIC COMPOUNDS USED AS ANTI-NEOPLASIC AGENTS OR CELL PROLIFERATION INHIBITORS CEREP (FR) 2008-09-12 WO disclosed