SCHEMBL4744705

SCHEMBL4744705

N#Cc1cnc(-c2cccs2)nc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
ABCG2 Q9UNQ0 1/20 0.41
KDM4E B2RXH2 8/20 0.41
FOS P01100 1/20 0.41
JUN P05412 1/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
ADORA2A P29274 2/20 0.40
ADORA1 P30542 2/20 0.40
PIM1 P11309 1/20 0.40
CYP3A4 P08684 2/20 0.39
CYP2E1 P05181 1/20 0.39
CYP2A6 P11509 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2B6 P20813 1/20 0.39
CHEK1 O14757 1/20 0.39
ALDH1A1 P00352 8/20 0.39
LMNA P02545 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10727341 0.82 CHEK1 (0.41) MEN1KMT2AKDM4EADORA2AADORA1
SCHEMBL1461854 0.79 MEN1 (0.47) MEN1KMT2AKDM4EADORA2AADORA1
SCHEMBL1031032 0.75 CSNK2A1 (0.41) MEN1KMT2AKDM4EFOSJUN
SCHEMBL436102 0.75 NPC1 (0.45) MEN1KMT2AKDM4ENFKB1NFKB2
SCHEMBL27933640 0.75 KDM4E (0.46) MEN1KMT2AKDM4EADORA2AADORA1
SCHEMBL8052677 0.75 KDM4E (0.46) MEN1KMT2AKDM4ECYP3A4CYP2E1
SCHEMBL219003 0.74 CYP3A4 (0.45) MEN1KMT2AKDM4ECYP3A4CYP2E1
SCHEMBL24786993 0.74 FOS (0.49) MEN1KMT2AKDM4EFOSJUN
SCHEMBL1003749 0.73 CYP19A1 (0.58) MEN1KMT2AKDM4ENFKB1NFKB2
SCHEMBL28423248 0.72 CYP3A4 (0.44) MEN1KMT2AKDM4ECYP3A4CYP2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008110891-A2 NEW HETEROCYCLIC COMPOUNDS ORCHID RESEARCH LABORATORIES LIMITED, (IN) 2008-09-18 WO claimed