SCHEMBL474522

SCHEMBL474522

CCN1C(=O)COc2ccc(C(O)(C(C)c3ccc(-c4ccc(C(=O)O)c(F)c4Cl)cc3)C(F)(F)F)cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
THRB P10828 1/20 0.37
SLC5A1 P13866 3/20 0.37
SLC5A2 P31639 3/20 0.37
HTT P42858 2/20 0.37
USP2 O75604 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
POLB P06746 2/20 0.36
KMO O15229 1/20 0.35
TSHR P16473 1/20 0.34
MAPT P10636 2/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
KMT2A Q03164 1/20 0.34
KDM4E B2RXH2 1/20 0.34
CYP3A4 P08684 3/20 0.33
CYP2D6 P10635 3/20 0.33
OPRK1 P41145 3/20 0.33
UTS2R Q9UKP6 3/20 0.33
BRD4 O60885 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474459 0.89 ALDH1A1 (0.40) ALDH1A1THRBSLC5A1SLC5A2HTT
SCHEMBL474631 0.89 ALDH1A1 (0.41) ALDH1A1THRBSLC5A1SLC5A2HTT
SCHEMBL474545 0.83 ALDH1A1 (0.42) ALDH1A1THRBSLC5A1SLC5A2HTT
SCHEMBL12163919 0.83 ALDH1A1 (0.42) ALDH1A1THRBSLC5A1SLC5A2HTT
SCHEMBL474334 0.82 ALDH1A1 (0.41) ALDH1A1THRBSLC5A1SLC5A2HTT
SCHEMBL12163929 0.82 ALDH1A1 (0.41) ALDH1A1THRBSLC5A1SLC5A2HTT
SCHEMBL474632 0.82 USP2 (0.42) ALDH1A1THRBSLC5A1SLC5A2HTT
SCHEMBL12163951 0.81 ALDH1A1 (0.41) ALDH1A1THRBSLC5A1SLC5A2HTT
SCHEMBL474540 0.81 ALDH1A1 (0.41) ALDH1A1THRBSLC5A1SLC5A2HTT
SCHEMBL12163950 0.81 ALDH1A1 (0.42) ALDH1A1THRBSLC5A1SLC5A2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed