SCHEMBL4745939

SCHEMBL4745939

COc1ccc(OC)c(CC(N)c2ccccc2)c1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.65
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
IDO1 P14902 2/20 0.51
ADRA1A P35348 1/20 0.51
TAAR1 Q96RJ0 1/20 0.51
HSD17B10 Q99714 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C19 P33261 1/20 0.49
AOC3 Q16853 1/20 0.47
TSPO P30536 1/20 0.46
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14042631 0.82 CYP1A2 (0.46) HTR2AMEN1KMT2ATAAR1CYP1A2
SCHEMBL23243766 0.82 ATM (0.54) MEN1KMT2AIDO1TAAR1CYP2D6
SCHEMBL29445352 0.82 ATM (0.54) MEN1KMT2AIDO1TAAR1CYP2D6
SCHEMBL23243765 0.82 ATM (0.54) MEN1KMT2AIDO1TAAR1CYP2D6
SCHEMBL31545209 0.79 HTR2A (1.00) HTR2AIDO1ADRA1ATAAR1
SCHEMBL1740902 0.79 HTR2A (1.00) HTR2AIDO1ADRA1ATAAR1
SCHEMBL1740903 0.79 HTR2A (1.00) HTR2AIDO1ADRA1ATAAR1
SCHEMBL3460220 0.79 HTR2A (1.00) HTR2AIDO1ADRA1ATAAR1
Hydrochloric Acid SCHEMBL29542459 0.78 HTR2A (0.97) HTR2AIDO1ADRA1ATAAR1
Hydrochloric Acid SCHEMBL3486527 0.78 HTR2A (0.97) HTR2AIDO1ADRA1ATAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123821-A1 4, 5-DIHYDRO-LH-IMIDAZOL-2-AMINE DERIVATIVES FOR USE IN THE TREATMENT OF RESPIRATORY, CARDIOVASCULAR, NEUROLOGICAL OR GASTROINTESTINAL DISORDERS ALBIREO AB (SE) 2008-10-16 WO claimed
WO-2008123821-A1 4, 5-DIHYDRO-LH-IMIDAZOL-2-AMINE DERIVATIVES FOR USE IN THE TREATMENT OF RESPIRATORY, CARDIOVASCULAR, NEUROLOGICAL OR GASTROINTESTINAL DISORDERS ALBIREO AB (SE) 2008-10-16 WO disclosed