SCHEMBL4746236

SCHEMBL4746236

O=C(c1ccc(Cl)cc1)c1c(F)cc(O)cc1F

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.59
SRD5A2 P31213 1/20 0.48
CNR1 P21554 1/20 0.46
CNR2 P34972 1/20 0.46
LMNA P02545 3/20 0.45
HTT P42858 3/20 0.45
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
HSD17B1 P14061 1/20 0.44
HSD17B2 P37059 1/20 0.44
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
CDK2 P24941 1/20 0.43
MAPT P10636 3/20 0.43
HPGD P15428 3/20 0.43
PTGS2 P35354 1/20 0.43
NPC1 O15118 1/20 0.43
NFKB1 P19838 1/20 0.43
RAB9A P51151 1/20 0.43
NFKB2 Q00653 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4743106 0.80 MAPK1 (0.58) MAPK1SRD5A2CNR1CNR2LMNA
SCHEMBL4746218 0.80 MAPK1 (0.63) MAPK1SRD5A2CNR1CNR2LMNA
SCHEMBL30396659 0.80 MAPK1 (0.63) MAPK1SRD5A2CNR1CNR2LMNA
SCHEMBL4743101 0.79 HPGD (0.64) CNR1LMNACDK2MAPTHPGD
SCHEMBL26231411 0.78 MAPK1 (0.46) MAPK1SRD5A2CNR1CNR2LMNA
SCHEMBL3446105 0.77 SRD5A2 (0.58) MAPK1SRD5A2CNR1CNR2LMNA
SCHEMBL26231301 0.75 HPGD (0.46) MAPK1SRD5A2LMNAHTTCES2
Hydroquinone SCHEMBL9777901 0.74 MAPK1 (1.00) MAPK1SRD5A2CNR1CNR2LMNA
Hydroquinone SCHEMBL10635396 0.74 MAPK1 (1.00) MAPK1SRD5A2CNR1CNR2LMNA
SCHEMBL333466 0.74 MAPK1 (1.00) MAPK1SRD5A2CNR1CNR2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008107320-A1 PIPERIDINE AND PIPERAZINE DERIVATIVES USED AS ANTI-NEOPLASIC AGENTS OR CELL PROLIFERATION INHIBITORS CEREP (FR) 2008-09-12 WO disclosed