SCHEMBL4746245

SCHEMBL4746245

O=C(CN1CCN(CCCCCOc2ccc(C(=O)c3ccc(Cl)cc3)cc2)CC1)NCc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.59
KCNA5 P22460 2/20 0.57
KDM4E B2RXH2 4/20 0.54
ALDH1A1 P00352 3/20 0.54
BCHE P06276 4/20 0.54
ACHE P22303 4/20 0.54
HRH3 Q9Y5N1 7/20 0.53
POLB P06746 1/20 0.52
RECQL P46063 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
HRH1 P35367 1/20 0.52
HTR7 P34969 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4746213 0.91 HRH4 (0.57) HRH4KCNA5KDM4EALDH1A1BCHE
SCHEMBL4747562 0.86 HRH3 (0.55) HRH4KCNA5HRH3MEN1KMT2A
SCHEMBL4743805 0.86 KDM4E (0.69) HRH4KDM4EALDH1A1BCHEACHE
SCHEMBL4745332 0.84 HRH3 (0.57) HRH4KCNA5HRH3MEN1KMT2A
SCHEMBL4746238 0.83 HRH3 (0.65) HRH4KDM4EALDH1A1HRH3MEN1
SCHEMBL4745346 0.82 HRH3 (0.51) HRH4KCNA5BCHEACHEHRH3
SCHEMBL4743288 0.81 HRH3 (0.56) HRH4KCNA5HRH3MEN1KMT2A
SCHEMBL4743111 0.81 HRH3 (0.56) HRH4KCNA5HRH3MEN1KMT2A
SCHEMBL4743293 0.80 MEN1 (0.56) HRH4KCNA5KDM4EALDH1A1HRH3
SCHEMBL4743806 0.79 TMEM97 (0.63) HRH4KDM4EALDH1A1BCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008107320-A1 PIPERIDINE AND PIPERAZINE DERIVATIVES USED AS ANTI-NEOPLASIC AGENTS OR CELL PROLIFERATION INHIBITORS CEREP (FR) 2008-09-12 WO claimed