SCHEMBL4747262

SCHEMBL4747262

CCOC(=O)[C@H](Cc1ccc2nc(-c3c(Cl)cccc3Cl)ccc2c1)NC(=O)OC(C)(C)C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 2/20 0.58
ITGAV P06756 1/20 0.58
CTSS P25774 5/20 0.45
CTSK P43235 5/20 0.45
CTSB P07858 3/20 0.45
ALDH1A1 P00352 4/20 0.43
MAPT P10636 3/20 0.43
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
GAA P10253 1/20 0.43
PKM P14618 1/20 0.43
ALOX12 P18054 1/20 0.43
CTSL P07711 1/20 0.43
PTPN1 P18031 1/20 0.42
SCN9A Q15858 1/20 0.39
TACR1 P25103 2/20 0.38
ACE P12821 1/20 0.38
KLK5 Q9Y337 1/20 0.38
DGAT1 O75907 1/20 0.38
ITGA4 P13612 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1030225 0.93 ITGB1 (0.59) ITGB1ITGAVCTSSCTSKCTSB
SCHEMBL3320795 0.93 ITGB1 (0.59) ITGB1ITGAVCTSSCTSKCTSB
SCHEMBL4627521 0.93 ITGB1 (0.59) ITGB1ITGAVCTSSCTSKCTSB
SCHEMBL4626858 0.90 ITGB1 (0.71) ITGB1ITGAVCTSSCTSKCTSB
SCHEMBL3315439 0.90 ITGB1 (0.71) ITGB1ITGAVCTSSCTSKCTSB
SCHEMBL3318595 0.90 ITGB1 (0.71) ITGB1ITGAVCTSSCTSKCTSB
SCHEMBL4625521 0.85 ITGB1 (0.49) ITGB1ITGAVCTSSCTSKCTSB
SCHEMBL3317515 0.85 ITGB1 (0.75) ITGB1ITGAVMAPTKDM4EITGA4
SCHEMBL4625325 0.84 CTSS (0.47) ITGB1ITGAVCTSSCTSKCTSB
SCHEMBL3315305 0.82 ITGB1 (0.52) ITGB1ITGAVCTSSCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008138592-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-11-20 WO disclosed
WO-2008125215-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-10-23 WO disclosed