SCHEMBL4747265

SCHEMBL4747265

CCC(c1ccc2nc(-c3c(Cl)cccc3Cl)ccc2c1)[C@H](NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.47
ITGAV P06756 1/20 0.47
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 3/20 0.40
HPGD P15428 3/20 0.40
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
THRB P10828 1/20 0.37
ABL1 P00519 1/20 0.37
HTT P42858 1/20 0.36
SUV39H2 Q9H5I1 2/20 0.35
CTSL P07711 1/20 0.34
EGFR P00533 1/20 0.34
TRPA1 O75762 1/20 0.34
GABRB1 P18505 1/20 0.34
GABRB2 P47870 1/20 0.34
S1PR3 Q99500 2/20 0.34
CA2 P00918 1/20 0.33
LCK P06239 1/20 0.33
ACSS2 Q9NR19 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1030227 0.89 ITGB1 (0.46) ITGB1ITGAVKDM4EALDH1A1HPGD
SCHEMBL3315439 0.80 ITGB1 (0.71) ITGB1ITGAVCTSL
SCHEMBL3318595 0.80 ITGB1 (0.71) ITGB1ITGAVCTSL
SCHEMBL4626858 0.80 ITGB1 (0.71) ITGB1ITGAVCTSL
SCHEMBL4747262 0.76 ITGB1 (0.58) ITGB1ITGAVKDM4EALDH1A1HPGD
SCHEMBL29231873 0.76 PPARG (0.50) KDM4EALDH1A1HPGDHTTTRPA1
SCHEMBL30192895 0.76 PPARG (0.50) KDM4EALDH1A1HPGDHTTTRPA1
SCHEMBL3320795 0.75 ITGB1 (0.59) ITGB1ITGAVCTSL
SCHEMBL1030225 0.75 ITGB1 (0.59) ITGB1ITGAVCTSL
SCHEMBL4627521 0.75 ITGB1 (0.59) ITGB1ITGAVCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008138592-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-11-20 WO disclosed
WO-2008125215-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-10-23 WO disclosed